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← ACTIVESRECORD A-18FAMILY MICROTUBULE INHIBITOR

Tirbanibulin

Tirbanibulin

Five days, then you stop. The shortest course in this register and the largest treatment difference after bimatoprost — for the photodamaged population every anti-ageing trial excluded.

THE TRIALLED STRENGTH, IN THE RANGE WE HAVE SEEN1% ——— 1%
1%

The marker is the strength the trials were actually run at. The bar is the span this register has recorded, approved and compounded together. Anything below the marker is a dose nobody has tested; anything above it is an assumption about a dose–response curve nobody has drawn.

IDENTITY & RATINGSA
INCITirbanibulin
FAMILYMicrotubule inhibitor
MOL. WEIGHT431.5 g/mol
REFERENCE CONC.1%
RANGE SEEN1 – 1%
STATUSPRESCRIPTION ONLY
ACTS ATEPIDERMIS
ONSET8 WK
STABILITYUNIT-DOSE PACKETS · SINGLE USE
TRIALS ON FILE2
IRRITATION INDEX8 / 10
STRATUM CORNEUMEPIDERMISDERMIS

The shaded band is the depth this molecule is understood to reach. Anything below it is out of scope, whatever the label says.

01

Mechanism

EVIDENCE GRADE A

Disrupts tubulin polymerisation in rapidly proliferating cells. Applied as a field treatment rather than lesion by lesion, so it acts on the subclinical damage around visible lesions as well as the lesions themselves.

HOUSE NOTES

  • Unit-dose packets remove the dosing judgement entirely — one packet, once a day, five days, with nothing left to over-apply.
  • The endpoint was complete clearance: no clinically visible lesions remaining, not fewer.
  • Local skin reactions are severe by the standards of this register — erythema worse than baseline in 91% of subjects — and they are the treatment working over a five-day course that then heals.
  • The face clears roughly twice as reliably as the scalp, and the label reports the two separately rather than pooling them.
  • Its trial population averaged 70 years old. Renova's excluded anyone with visible actinic keratosis, which is the same population seen from the other side.

MEASURED ENDPOINTS

Complete (100%) lesion clearance+42%
8 WKREF-29
Erythema worse than baseline-57%
1 WKREF-30

SUPPORTING RECORDS

  • Double-blind, vehicle-controlled, five-day course; average subject age 70, range 45 to 96

    N=351 · 8 WK · DOUBLE-BLIND

  • Investigator-graded local skin reactions in the treatment area, pooled across both Phase 3 trials

    N=702 · 8 WK · DOUBLE-BLIND

02

Layering

CONFLICTS & PAIRINGS
DO NOT LAYER
  • Occlusion after application
  • Skin not yet healed from prior treatment or surgery
  • Eyes, mouth and nostrils
PAIRS WITH
  • Daily sunscreen, permanently, afterwards
03

Reviewed in

1 REVIEW
EVERY FIGURE HERE RESOLVES TO A RECORD IN THE EVIDENCE REGISTER. NOT MEDICAL ADVICE.
THE DRAW · NO. 01

Win a year of
prescription skincare

One reader gets a 12 months CoreAge Rx derm plan — the compounded, physician-reviewed subscription we take apart in the register. Worth $780. Leave an address and you are entered.

PRIZE
12 MONTHS OF COREAGE RX
VALUE
$780 — $64.99/MO × 12
ENTRY
ONE EMAIL ADDRESS

VALUE IS THE PUBLISHED $64.99/MONTH SUBSCRIPTION PRICE OVER TWELVE MONTHS, AS RECORDED IN R-10. NO PURCHASE NECESSARY. WE REVIEW COREAGE RX — WE DO NOT SELL IT.

DEPTH 000%
THE DRAW · ONE READER

Win a year of
prescription skincare

One reader gets a 12 months CoreAge Rx derm subscription — compounded, physician-reviewed, delivered. The plan we score in the register.

VALUE$780
TERM12 MONTHS$64.99/MO × 12

VALUE IS THE PUBLISHED $64.99/MONTH SUBSCRIPTION PRICE OVER TWELVE MONTHS, AS RECORDED IN R-10. NO PURCHASE NECESSARY. WE REVIEW COREAGE RX — WE DO NOT SELL IT.